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Product Detail

  • Apalutamide
  • Apalutamide
  • Apalutamide
  • Apalutamide


  • CAS No.956104-40-8:
  • Molecular Formula:C21H15F4N5O2S:
  • Molecular Weight:477.4:
  • Reference Standard:In-house:
  • Documentation:TP:
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Product Description

Apalutamide is a small molecule and androgen receptor (AR) antagonist with potential antineoplastic activity. Apalutamide binds to AR in target tissues thereby preventing androgen-induced receptor activation and facilitating the formation of inactive complexes that cannot be translocated to the nucleus. This prevents binding to and transcription of AR-responsive genes. This ultimately inhibits the expression of genes that regulate prostate cancer cell proliferation and may lead to an inhibition of cell growth in AR-expressing tumor cells.

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